BIM-23627

H-p-Chloro-Phe-D-Cys-β-(2-pyridyl)-Ala-Trp-Lys-Val-Cys-2-Nal-NH₂ (Disulfide bond)

Product Number: 4041642

CAS Number: 429619-37-4

€ 240.80 – € 428

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Product Description

The somatostatin antagonist BIM 23627 selectively bound with high affinity to the human somatostatin receptor subtype 2 (hsst2), but was completely inactive in stimulating intracellular calcium mobilization. The IC₅₀ values of BIM 23627 to the five human somatostatin receptor subtypes were 2757 nM (hsst1), 6.4 nM (hsst2), 44 nM (hsst3), 423 nM (hsst4), and 86.5 nM (hsst5).

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Peptides in cancer research
Highly potent and subtype selective ligands derived by N-methyl scan of a somatostatin antagonist.

W.G.Rajeswaran et al., J. Med. Chem., 44, 1305 (2001)

Salt form: Trifluoroacetate

Molecular weight: 1161.85

Chemical Formula: C₅₈H₆₉ClN₁₂O₈S₂

Storage Temperature: < -15°C

Source: Synthetic

Old Product Number: H-5886

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