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Availability: In stock

H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-Lys-tBu-Gly-Cys-2-Nal-NH₂ trifluoroacetate salt (Disulfide bond)

4044525

Product No. Pack Size Available ADS InfoAnalytical Data Sheet Unit Price Online Order Price Qty
4044525.0500 0.5 mg Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 137.00
CHF 127.41 (7%)
4044525.1000 1 mg Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 232.00
CHF 215.76 (7%)
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Details

PRL2915, Cpa-D-Cys-Pal-D-Trp-Lys-Tle-Cys-Nal-amide, highly potent human somatostatin subtype 2 receptor (hsst2) antagonist with a Ki of 12 nM. Ki values for the other subtypes were >1000 nM for hsst1, 100 ± 57 nM for hsst3, 895 nM for hsst4, and 520 nM for hsst5, respectively. No agonist activity was found when tested alone at concentrations up to 10 µM. In a rat pituitary growth hormone in vitro antagonist assay versus somatostatin-14 (1nM) the somatostatin octapeptide analog PRL2915 exhibited an IC₅₀ value of 1.8 nM.
Catalog Number H-6056
Synonyms PRL-2915
Molecular Formula C₅₉H₇₁ClN₁₂O₈S₂
Relative Molecular Mass 1175.87
CAS Registry Number [209006-18-8] net
Source Synthetic
Storage Conditions -20 ± 5 °C