Return to Previous Page
Details
This synthetic somatostatin analog is selective for the human somatostatin receptor subtype 5 (hsst5) with a binding affinity similar to somatostatin-28. Its Kd +/-SEM values for hsst1, hsst2, hsst3, hsst4, and hsst5 are 1200 nM, 23.5 +/- 3.92 nM, 11.05 +/- 1.03 nM, > 1000 nM, and 0.61 +/- 0.36 nM, respectively. Due to its selectivity it might prove to be useful for evaluating hsst5-mediated responses.
Catalog Number
H-5648
Synonyms
(N-Me-D-Trp⁴)-Octreotate amide, (N-Me-D-Trp⁴,Thr⁸)-Octreotide amide
Molecular Formula
C₅₀H₆₇N₁₁O₁₀S₂
Relative Molecular Mass
1046.28
CAS Registry Number
340821-13-8
Source
Synthetic
Storage Conditions
-20 ± 5 °C
Application
Cancer Research
Links / Documents:
Brochures:
