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4034493

Availability: In stock

(d(CH₂)₅¹,Tyr(Me)²,Orn⁸)-Oxytocin trifluoroacetate salt

4034493

Product No. Pack Size Available ADS InfoAnalytical Data Sheet List Price Online Order Price Qty
4034493.0001 1 Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 232.00
CHF 215.76 (7%)
4034493.0005 5 Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 924.00
CHF 859.32 (7%)

Details

Potent oxytocin antagonist with a pA₂ value of 7.35 ± 0.08. (d(CH₂)₅¹,Tyr(Me)²,Orn⁸)-Vasotocin has been used to support the hypothesis that pituitary secretion of oxytocin is associated with coactivation of centrally projecting brain oxytocin pathways, some of which are causally related to the induced inhibition of food intake. Furthermore, this compound competitively inhibited arginine vasotocin (AVT) contractions without affecting AVT efficacy.
APC Number 66-0-16
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Bachem product citations

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