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Availability: In stock

Tertiapin
H-Ala-Leu-Cys-Asn-Cys-Asn-Arg-Ile-Ile-Ile-Pro-His-Met-Cys-Trp-Lys-Lys-Cys-Gly-Lys-Lys-NH₂
(Disulfide bonds between Cys³ and Cys¹⁴/Cys⁵ and Cys¹⁸)

4031297

Product No. Pack Size Available ADS InfoAnalytical Data Sheet Unit Price Online Order Price Qty
4031297.0500 0.5 mg Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 420.00
CHF 390.60 (7%)
4031297.1000 1 mg Ships within 3-5 business days  
CHF 735.00
CHF 683.55 (7%)
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Details

Tertiapin (TPN), a potent inhibitor of the inward-rectifier K⁺ channels, blocked a G-protein-gated channel (GIRK1/4) and the ROMK1 channel with nanomolar affinities, however a closely related channel, IRK1, was insensitive to tertiapin. Thus, tertiapin will be a powerful ligand for purifying functional channels as well as for screening pharmaceutical agents against these channels.
Catalog Number N-1745
One Letter Code ALCNCNRIIIPHMCWKKCGKK -NH₂
Molecular Formula C₁₀₆H₁₇₆N₃₄O₂₃S₅
Relative Molecular Mass 2455.11
CAS Registry Number [58694-52-3]
Source Synthetic
Storage Conditions -20 ± 5 °C
Keywords Channel-blocking peptide from bee venom
Areas of Interest Ion Channel Modulating Agents