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Myristoyl-(Lys¹²·²⁷·²⁸)-VIP-Gly-Gly-Thr (free acid) trifluoroacetate salt
Myristoyl-His-Ser-Asp-Ala-Val-Phe-Thr-Asp-Asn-Tyr-Thr-Lys-Leu-Arg-Lys-Gln-Met-Ala-Val-Lys-Lys-Tyr-Leu-Asn-Ser-Ile-Lys-Lys-Gly-Gly-Thr-OH trifluoroacetate salt

H-7292

Product No. Pack Size Available ADS InfoAnalytical Data Sheet Unit Price Online Order Price Qty
H-7292.0500 0.5 mg Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 260.00
CHF 241.80 (7%)
H-7292.1000 1 mg Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 450.00
CHF 418.50 (7%)
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Details

PG 99-465 is a high affinity, selective VPAC2 receptor antagonist. It exhibited a 100-fold preference for the VPAC2 over the VPAC1 receptor. The compound showed partial agonistic activity on the VPAC1 receptor and was inactive on the VPAC2 receptor transfected in CHO cells, as well as on naturally expressed human VPAC2 receptors in the SUP T1 cell line.
Dickson et al. observed an agonistic effect of PG99-465 on the human VPAC1 and PAC1 receptors. When applied singly, PG99-465 increased [cAMP](i) at all three hVPAC/PAC receptor subtypes.
Item Number 4037992
Synonyms PG 99-465
Molecular Formula C₁₇₁H₂₈₃N₄₅O₄₇S
Relative Molecular Mass 3753.47
Source Synthetic
Storage Conditions -20 ± 5 °C