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H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-Lys-tBu-Gly-Cys-2-Nal-NH₂ trifluoroacetate salt (Disulfide bond)

H-6056

Product No. Pack Size Available ADS InfoAnalytical Data Sheet Unit Price Online Order Price Qty
H-6056.0500 0.5 mg Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 134.00
CHF 124.62 (7%)
H-6056.1000 1 mg Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 227.00
CHF 211.11 (7%)
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Details

PRL2915, Cpa-D-Cys-Pal-D-Trp-Lys-Tle-Cys-Nal-amide, highly potent human somatostatin subtype 2 receptor (hsst2) antagonist with a Ki of 12 nM. Ki values for the other subtypes were >1000 nM for hsst1, 100 ± 57 nM for hsst3, 895 nM for hsst4, and 520 nM for hsst5, respectively. No agonist activity was found when tested alone at concentrations up to 10 µM. In a rat pituitary growth hormone in vitro antagonist assay versus somatostatin-14 (1nM) the somatostatin octapeptide analog PRL2915 exhibited an IC₅₀ value of 1.8 nM.
Item Number 4044525
Synonyms PRL-2915
Molecular Formula C₅₉H₇₁ClN₁₂O₈S₂
Relative Molecular Mass 1175.87
CAS Registry Number [209006-18-8] net
Source Synthetic
Storage Conditions -20 ± 5 °C