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Availability: In stock

BQ-610
Azepane-1-carbonyl-Leu-D-Trp(For)-D-Trp-OH

H-4914

Product No. Pack Size Available ADS InfoAnalytical Data Sheet Unit Price Online Order Price Qty
H-4914.0500 0.5 mg Ships within 3-5 business days  
CHF 95.00
CHF 88.35 (7%)
H-4914.1000 1 mg Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 158.00
CHF 146.94 (7%)
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Details

BQ-610 is a very potent ET-A receptor antagonist which is about 30000 times more selective for ET-A receptors than for ET-B receptors. Furthermore, it has been found that BQ-610 strongly antagonizes ET-1 induced concentration in porcine coronary artery with a pA₂ value of 8.2.
Item Number 4034542
APC Number 88-2-32
Molecular Formula C₃₆H₄₄N₆O₆
Relative Molecular Mass 656.78
CAS Registry Number [141595-53-1]
Source Synthetic
Storage Conditions -20 ± 5 °C
Keywords Endothelin antagonist. BQ610 binds to the ET-A receptor with IC₅₀ 20 nM.