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Availability: In stock

BQ-788
N-cis-2,6-Dimethylpiperidinocarbonyl-β-tBu-Ala-D-Trp(1-methoxycarbonyl)-D-Nle-OH

H-2492

Product No. Pack Size Available ADS InfoAnalytical Data Sheet Unit Price Online Order Price Qty
H-2492.0001 1 mg Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 268.00
CHF 249.24 (7%)
H-2492.0005 5 mg Ships within 1 business day ADSExemplary Data Sheet of a current available lot.
CHF 1'071.00
CHF 996.03 (7%)
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Details

In vitro, BQ-788 potently and competitively inhibited ¹²⁵I-labeled ET-1 binding to ET-B receptors on human Girardi heart cells (IC₅₀= 1.2 nM). However, BQ-788 only poorly inhibited ET-1 binding to ET-A receptors on human neuroblastoma cell line SK-N-MC cells (IC₅₀= 1300 nM). Thus the ET-B receptor antagonist BQ788 may be considered as a powerful tool for investigating the role of ET in physiological and pathological processes.
Item Number 4026108
Molecular Formula C₃₄H₅₁N₅O₇
Relative Molecular Mass 641.81
CAS Registry Number [173326-37-9]
Source Synthetic
Storage Conditions -20 ± 5 °C
Keywords Endothelin antagonist